N
H
HO
H
2
N
N
H
HO
H
2
N
N
H
HO
H
2
N
SpiroperidolSpiperone
Iodocyanopindolol(5-HT 1B)
Rauwolscine(5-HT 1D)
8-OH-DPAT
8-OH-DPATLSD5-CT
GIRK
Ca
2+
Ca
2+
5-HT1A
5-HT1B-1F
5-HT5
5-HT4
5-HT6
5-HT7
cAMP
PKA
Raf
PKC
MEK
MAPK
ERK1/2
AC
ATP
p90 RSK2
CREB
CRE
PIP
2
IP
3
DAG
BDNF
β-arr
γ
β
γ
β
γ
β
αi/0
αs
LSD
Mesulergine
Serotonylation of Rab Proteins
5-HT2A
5-HT2B
5-HT2C
SERT
γ
PLCβ
PLCγ
PH
Src
PLA
2
PLD
Arachidonic Acid
Phosphatidylcholine
Phosphatidic Acid
RhoA-GEF
RhoA
γ
β
β
αq/11
α12/13
NF-κB
PI3K
Akt
PKA
ERK1/2
MAPK
MEK
Raf
Ras
5-HT Receptor AntagonistsClozapineOlanzapineKetanserin5-HT Receptor AgonistsPrucaloprideWAY-100635 Eletriptan
Pan-MEK InhibitorsTrametinibU0126-EtOHPD184352Selective MEK InhibitorsSelumetinib (MEK1)BIX 02189 (MEK5)
PKA InhibitorsA-674563H 89AT13148
Pan-Akt InhibitorsMK-2206PerifosineGSK690693Selective Akt InhibitorsA-674563 (Akt1)CCT128930 (Akt2)
Rho Family InhibitorsZoledronic AcidNSC 23766EHop-016ZCL278
PKA InhibitorsA-674563H 89AT13148
ERK InhibitorsSCH772984XMD8-92FR 180204GDC-0994
cAMP ActivatorForskolin
P
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GIRK
Mesulergine
SERT
Serotonylation of Rab Proteins
Arachidonic Acid
Phosphatidylcholine
Phosphatidic Acid
8-OH-DPAT
Spiroperidol
Spiperone
Iodocyanopindolol
(5-HT 1B)
Rauwolscine
(5-HT 1D)
8-OH-DPAT
LSD
5-CT
LSD
Ca
Ca
2+
2+
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2
2
3
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Notes:
1:Clickable
2:Unclickable