TGFβ
ROCK
PAK
c-Abl
PKC
Smad3
Smad2
Smad4
Smad4
Smad2
Smad3/4
Smad2/4
Ras
MEKs
ERK1/2
Smad7
Smad6
Transcription
Actin PolymerizationStress Fibers
Cell Adhesion
TumorSuppression
Cell Growth
SBE
LIMK
PI3K/AktPathway
MAPKPathway
CDC42
Apoptosis
Angiogenesis
P300
CBP
Pan-ROCK InhibitorsY-27632ThiazovivinFasudilRipasudilSelective ROCK InhibitorKD025 (ROCK2)
PAK InhibitorsFRAX597PF-3758309IPA-3
Bcr-Abl InhibitorsPonatinibImatinibNilotinibDegrasynAsciminib
Pan-TGF-beta/Smad InhibitorsLDN-193189K02288Selective TGF-beta/Smad InhibitorsSB431542 (ALK5)Galunisertib (TGF-βRI)
Pan-TGF-beta/Smad InhibitorsLDN-193189K02288Selective TGF-beta/Smad InhibitorsSB431542 (ALK5)Galunisertib (TGF-βRI)
Ras InhibitorsARS-1620ARS-853KRpep-2dAMG510BAY-293
Pan-MEK InhibitorsTrametinibPD0325901SelumetinibU0126-EtOHPD98059Selective MEK InhibitorsCobimetinib (MEK1)BIX 02189 (MEK5)
P
Apoptosis
Angiogenesis
PI3K/Akt
Pathway
MAPK
Pathway
Cell Adhesion
Transcription
Cell Growth
Actin Polymerization
Stress Fibers
Tumor
Suppression
SBE
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1:Clickable
2:Unclickable